Skip to main navigation menu Skip to main content Skip to site footer

Articles

Vol. 1 (2023): KolaDaisi University Journal of Applied Sciences

Oxidative Stress-Induced Spermiotoxicity of Ciprofloxacin: An In Vitro Study

DOI:
https://doi.org/10.5281/zenodo.17372122
Submitted
October 22, 2025
Published
August 24, 2023

Abstract

Infertility can primarily result from oxidative stress induced by the use of various drugs including known antibiotics.
This study investigated dose and time-dependent effect of Ciprofloxacin on antioxidant status, sperm motility, viability and morphological characteristics of semen from sexually mature boar. Semen was incubated with Ciprofloxacin at 5.4 μg/ml, 54 μg/ml and 540 μg/ml for 4 hours at 37oC and sperm characteristics were monitored at 2-hour intervals.
Antioxidant status was assessed after the incubation period by estimation of reduced glutathione levels, and activities of glutathione S-transferase, glutathione peroxidase, superoxide dismutase and catalase. The extent of lipid peroxidation and hydrogen peroxide generation were also determined. Ciprofloxacin induced oxidative stress in boar semen in a dose-dependent manner with a significant increase (p < 0.05) in reduced glutathione levels, and activities of glutathione-S-transferase, glutathione peroxidase, and catalase as well as malondialdehyde and hydrogen peroxide levels when compared with the control. However, when compared with the control, there was a significant (p < 0.05) dose-dependent decline in the activity of SOD. Assessment of sperm characteristics revealed a decline in motility, 2 hours post-treatment with all doses of Ciprofloxacin which became significant in the 4th hour. Semen incubation with Ciprofloxacin also increased the number of abnormal sperm cells while decreasing viability in a time-dependent manner. Overall, these results show that Ciprofloxacin caused enhancement of free radicals and alterations in activities of antioxidant enzymes with a resultant deterioration in sperm motility, viability and morphology.